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Nefopam Mechanism — FRCA Final MCQ

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ModeratePain MedicineNefopam MechanismFRCA Final

Nefopam mechanism of action is:

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Correct answer: AGABA modulation

Nefopam inhibits serotonin/noradrenaline/dopamine reuptake and modulates sodium channels. Non-opioid, no respiratory depression, ~equivalent to morphine 10 mg oral.

Reference: BNF – 2025 – Nefopam