ergometrine maleate · Medicine question

How is ergometrine maleate metabolised in the body?

iatroX medicinesPublished 8 November 2026

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Ergometrine maleate is mainly metabolised in the liver by hydroxylation and glucuronic acid conjugation, possibly also by N-demethylation, and is a substrate for CYP3A4 enzymes.

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Ergometrine Injection BP 0.05% w/vhameln pharma ltd · emc · SmPC §5.2 Pharmacokinetic properties · Version 7Document updated 5 May 2026

Sources checked 8 November 2026

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